Caeruleanone A, a Rotenoid with a New Arrangement of the D-Ring from the Fruits of Millettia caerulea

نویسندگان

  • Lynette Bueno Pérez
  • Li Pan
  • Ulyana Muñoz Acuña
  • Jie Li
  • Hee-Byung Chai
  • Judith C. Gallucci
  • Tran Ngoc Ninh
  • Esperanza J. Carcache de Blanco
  • Djaja D. Soejarto
  • A. Douglas Kinghorn
چکیده

Caeruleanone A (1), a novel rotenoid with an unprecedented arrangement of the D-ring, was isolated with another two new analogues, caeruleanones B (2) and C (3), together with 11 known rotenoids from the fruits of Millettia caerulea. The structures of the new compounds were determined by spectroscopic data analysis, with that of 1 being confirmed by single-crystal X-ray diffraction. Compounds 2 and 3 displayed potent mitochondrial transmembrane potential inhibitory and quinone reductase induction activities.

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عنوان ژورنال:

دوره 16  شماره 

صفحات  -

تاریخ انتشار 2014